| HS Code | 268638 |
| Product Name | Lifitegrast Intermediates Pharma Grade API for Tablet / Capsule / Granule / Injection, Oral & Injectable |
| Product Type | Pharma grade API and intermediate |
| Cas Number | 1025967-78-5 |
| Molecular Formula | C29H24Cl2N2O7S |
| Molecular Weight | 615.48 g/mol |
| Iupac Name | (2S)-2-[[2-(1-benzofuran-6-carbonyl)-5,7-dichloro-1,2,3,4-tetrahydroisoquinoline-6-carbonyl]amino]-3-(3-methylsulfonylphenyl)propanoic acid |
| Synonyms | Lifitegrast; Xiidra; SAR 1118; Lifitegrastum |
| Drug Class | Lymphocyte function-associated antigen-1 (LFA-1) antagonist; integrin inhibitor |
| Therapeutic Category | Ophthalmic agent; dry eye disease treatment |
| Mechanism Of Action | Blocks LFA-1 binding to ICAM-1, reducing T-cell-mediated inflammation |
| Chemical Family | Isoquinoline derivative; benzofuran derivative |
| Appearance | White to off-white crystalline powder |
| Purity | >=98.0% (HPLC) |
| Assay | 98.0% to 102.0% (anhydrous basis) |
| Grade | Pharma Grade; GMP |
| Optical Purity | Single S-enantiomer |
| Solubility | Soluble in DMSO and methanol; aqueous solubility is pH-dependent |
| Storage Conditions | Store in a cool, dry, well-ventilated area protected from light and moisture; recommended 2-8 C |
| Shelf Life | 24 to 36 months when stored properly |
| Dosage Forms | Tablet, capsule, granule, injection |
| Route Of Administration | Oral, injectable; ophthalmic for approved lifitegrast |
| Packaging | 1 kg, 5 kg, 10 kg, 25 kg in fiber drums with double polyethylene bags |
| Hs Code | 29349990 |
| Use | Treatment of dry eye disease |
| Residual Solvents | Controlled per ICH guidelines |
| Heavy Metals | Controlled per ICH guidelines |
As an accredited Lifitegrast Intermediates Pharma Grade API for Tablet / Capsule / Granule / Injection, Oral & Injectable factory, we enforce strict quality protocols—every batch undergoes rigorous testing to ensure consistent efficacy and safety standards.
| Packing | |
| Shipping | |
| Storage |
Competitive Lifitegrast Intermediates Pharma Grade API for Tablet / Capsule / Granule / Injection, Oral & Injectable prices that fit your budget—flexible terms and customized quotes for every order.
For samples, pricing, or more information, please contact us at +8615365186327 or mail to admin@ascent-chem.com.
We will respond to you as soon as possible.
Tel: +8615365186327
Email: admin@ascent-chem.com
Flexible payment, competitive price, premium service - Inquire now!
